Paralog-dependent isogenic cell assay cascade generates highly selective SLC16A3 inhibitors

Dvorak V, Casiraghi A, Colas C, Koren A, Tomek T, Offensperger F, Rukavina A, Tin G, Hahn E, Dobner S, Frommelt F, Boeszoermenyi A, Bernada V, Hannich JT, Ecker GF, Winter GE, Kubicek S and Superti-Furga G

Cell Chemical Biology, 2023

doi:10.1016/j.chembiol.2023.06.029.

E3-specific degrader discovery by dynamic tracing of substrate receptor abundance.

Hanzl A, Barone E, Bauer S, Yue H, Nowak RP, Hahn E, Pankevich EV, Koren A, Kubicek S, Fischer ES, Winter GE

Journal of the American Chemical Society, 2023

doi:10.1021/jacs.2c10784.

Publisher correction: rational discovery of molecular glue degraders via scalable chemical profiling.

Mayor-Ruiz C, Bauer S, Brand M, Kozicka Z, Siklos M, Imrichova H, Kaltheuner IH, Hahn E, Seiler K, Koren A, Petzold G, Fellner M, Bock C, Muller AC, Zuber J, Geyer M, Thoma NH, Kubicek S, Winter GE

Nature chemical biology, 2021

doi:10.1038/s41589-021-00735-4.

Rational discovery of molecular glue degraders via scalable chemical profiling.

Mayor-Ruiz C, Bauer S, Brand M, Kozicka Z, Siklos M, Imrichova H, Kaltheuner IH, Hahn E, Seiler K, Koren A, Petzold G, Fellner M, Bock C, Müller AC, Zuber J, Geyer M, Thomä NH, Kubicek S, Winter GE

Nature chemical biology, 2020

doi:10.1038/s41589-020-0594-x.