The ChEMBL Database in 2023: a drug discovery platform spanning multiple bioactivity data types and time periods.

Zdrazil B, Felix E, Hunter F, Manners EJ, Blackshaw J, Corbett S, de Veij M, Ioannidis H, Lopez DM, Mosquera JF, Magarinos MP, Bosc N, Arcila R, Kizilören T, Gaulton A, Bento AP, Adasme MF, Monecke P, Landrum GA, Leach AR.

Nucleic Acids Res, 2024

doi:10.1093/nar/gkad1004.

eTRANSAFE: data science to empower translational safety assessment.

Sanz F, Pognan F, Steger-Hartmann T, Díaz C, Asakura S, Amberg A, Bécourt-Lhote N, Blomberg N, Bosc N, Briggs K, Bringezu F, Brulle-Wohlhueter C, Brunak S, Bueters R, Callegaro G, Capella-Gutierrez S, Centeno E, Corvi J, Cronin MTD, Drew P, Duchateau-Nguyen G, Ecker GF, Escher S, Felix E, Ferreiro M, Frericks M, Furlong LI, Geiger R, George C, Grandits M, Ivanov-Draganov D, Kilgour-Christie J, Kiziloren T, Kors JA, Koyama N, Kreuchwig A, Leach AR, Mayer MA, Monecke P, Muster W, Nakazawa CM, Nicholson G, Parry R, Pastor M, Piñero J, Oberhauser N, Ramírez-Anguita JM, Rodrigo A, Smajic A, Schaefer M, Schieferdecker S, Soininen I, Terricabras E, Trairatphisan P, Turner SC, Valencia A, van de Water B, van der Lei JL, van Mulligen EM, Vock E, Wilkinson D.

Nat Rev Drug Discov, 2023

doi:10.1038/d41573-023-00099-5.

Illuminating the druggable genome through patent bioactivity data.

Magariños MP, Gaulton A, Félix E, Kiziloren T, Arcila R, Oprea TI, Leach AR.

PeerJ, 2023

doi:10.7717/peerj.15153.

Illuminating the Druggable Genome through Patent Bioactivity Data

Magariños MP, Gaulton A, Félix E, Kizilören T, Arcila R, Oprea T, Leach AR.

2022

doi:10.1101/2022.07.15.500187.